Identifying New Drug Targets for Potent Phospholipase D Inhibitors: Combining Sequence Alignment, Molecular Docking, and Enzyme Activity/Binding Assays

  • Helene Djakpa
  • , Aditya Kulkarni
  • , Scheneque Barrows-Murphy
  • , Greg Miller
  • , Weihong Zhou
  • , Hyejin Cho
  • , Béla Török
  • , Kimberly Stieglitz

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Pages (from-to)714-729
Number of pages16
JournalChemical Biology and Drug Design
Volume87
Issue number5
DOIs
StatePublished - May 1 2016

ASJC Scopus Subject Areas

  • Biochemistry
  • Molecular Medicine
  • Pharmacology
  • Drug Discovery
  • Organic Chemistry

Keywords

  • bioinformatics
  • biological screening
  • chemical biology
  • drug design
  • structural biology

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